Skip to main content

Table 2 List of VEGF Inhibitors

From: Nanoparticle mediated targeting of VEGFR and cancer stem cells for cancer therapy

Agent

Class

Target

References

Bevacuzimab

MAB

VEGF-A

[17, 18]

IMC-1121B

MAB

VEGFR-2

[19]

CDP-791

DiFabPEG

VEGFR-2

[20]

CEP-7055

TKI

VEGFR-1,2,3

[20]

PTK-787

TKI

VEGFR-1,2

[21]

AEE788

TKI

VEGFR-2, EGFR

[22]

ZD6474

TKI

VEGFR-1,2,3, EGFR

[23]

AG013736

TKI

VEGFR-1,2

[24]

AZD2171

TKI

VEGFR-1,2

[25]

SUO11248

TKI

VEGFR-1,2, PDGFR

[26]

CP-547,632

TKI

VEGFR-1,2

[27]

GW786024

TKI

VEGFR-1,2,3

[28]

Bay 93-4006

TKI

VEGFR-1,2, PDGFR

[29]

AMG 706

TKI

VEGFR-1,2,3

[30]